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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2058 | Palosuran | ACT-058362 | GPR |
Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor. | |||
T23323 | SB 611812 | Neurotensin Receptor | |
SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease. | |||
T22476 | (±)-AC 7954 hydrochloride | Neurotensin Receptor | |
(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator. | |||
T37527L | [Orn8]-Urotensin II acetate | GPR | |
[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors. | |||
T27328 | FL104 | FL-104,FL 104 | GPR |
FL104 is a potent agonist of small-molecule urotensin II receptor, pEC50= 7.11. | |||
TP1737L | Urotensin II (114-124), human acetate | Urotensin II (114-124), human acetate(251293-28-4 free base) | GPR |
Urotensin II (114-124), human acetate is an 11-amino acid residue peptide, is a potent vasoconstrictor and agonist for the orphan receptor GPR14. | |||
TP1928L1 | [Orn5]-URP acetate | [Orn5]-URP acetate(782485-03-4 free base) | GPR |
[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity. | |||
TP2104L | UFP 803 acetate | Neurotensin Receptor | |
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist. | |||
TP2106L | Urantide acetate(669089-53-6 free base) | Neurotensin Receptor | |
Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced ... | |||
TP1199L | Urotensin I acetate (83930-33-0 Free base) | CRFR | |
Urotensin I acetate, a CRF-like neuropeptide, acts as an agonist of CRF receptor with pEC50s of 11.46, 9.36 and 9.85 for human CRF1, human CRF2 and rat CRF2α receptors in CHO cells, and Kis of 0.4, 1.8, and 5.7 nM for hC... | |||
T12848 | SB-657510 | Others , Neurotensin Receptor | |
SB-657510 is a urotensin II (UII) receptor (UT) antagonist. The Ki values of UT for human, monkey, cat, rat and mouse were 61, 17, 30, 65 and 56 nM, respectively. SB-657510 plays an anti-inflammatory role by inhibiting U... | |||
T23326 | SB 706375 | Others | |
urotensin-II (UT) receptor antagonist | |||
T22815 | GSK 1562590 hydrochloride | Others | |
urotensin II (UT) receptor antagonist | |||
T28692 | SB-436811 | SB 436811 | |
SB-436811 is an antagonist of human urotensin-II receptor. | |||
T26542 | AC-7954 | ||
AC-7954 is a potent and efficacious agonist of urotensin II receptor. | |||
T71642 | GSK-1562590 | ||
GSK-1562590 is a urotensin-II receptor antagonist. | |||
T27441 | GSK 1440115 | GSK1440115,GSK-1440115 | |
GSK 1440115, an orally active urotensin II receptor antagonist, is used to treat asthma. | |||
T36729 | Urotensin II (goby) (trifluoroacetate salt) | ||
Urotensin II is a peptide vasoconstrictor and agonist of the urotensin (UT) receptor (Ki= 2.06 nM for the human recombinant receptor expressed in HEK293 cells).1It stimulates intracellular calcium mobilization in HEK293 ... | |||
TP1737 | Urotensin II (114-124), human | ||
Urotensin II (114-124), human, is an 11-amino acid residue peptide that exhibits strong vasoconstrictor activity and acts as an agonist for the orphan receptor GPR14. | |||
TP1415 | Urotensin II (114-124), human TFA | ||
Urotensin II (114-124), human TFA, is an 11-amino acid residue peptide with a strong vasoconstrictor effect. This compound acts as an agonist for the orphan receptor GPR14. |